Compare Peptides

Select any two compounds for a side-by-side comparison of mechanism, uses, risks, and FDA regulatory status.

Popular comparisons

GHRP-2

Growth Hormone Releasing Peptide-2, Pralmorelin

Unregulated
Growth Hormone Secretagogue

Hexarelin

Examorelin, His-D-2-MeTrp-Ala-Trp-D-Phe-Lys-NH2

Category 1
Growth Hormone Secretagogue
Overview

A synthetic hexapeptide growth hormone secretagogue that stimulates GH release through the ghrelin receptor. Considered one of the most potent GHRPs available, producing stronger GH pulses than GHRP-6 but with more appetite stimulation than ipamorelin. Widely used in anti-aging and performance contexts.

A synthetic hexapeptide growth hormone secretagogue and one of the most potent GH-releasing peptides known. Stimulates GH release more strongly than most other GHS peptides, but also has significant effects on cortisol and prolactin.

Mechanism of Action

Binds to the growth hormone secretagogue receptor (GHS-R1a / ghrelin receptor) in the anterior pituitary, triggering GH release. Also stimulates appetite through hypothalamic ghrelin pathways. Produces a robust GH pulse that synergizes with GHRH analogs like CJC-1295 or sermorelin.

Binds to ghrelin receptors (GHS-R1a) in the pituitary and hypothalamus, triggering strong GH release. Also has direct cardioprotective effects independent of GH, including protection against ischemia-reperfusion injury. Activates the CD36 receptor in cardiac tissue.

Common Uses
  • Growth hormone optimization
  • Muscle growth and recovery
  • Anti-aging protocols
  • Improved sleep quality
  • Fat loss (via elevated GH)
  • Growth hormone optimization
  • Muscle mass and strength
  • Fat loss
  • Cardiac protection (emerging research)
  • Recovery from injury
Known Risks
  • Increased appetite and hunger
  • Water retention
  • Elevated cortisol and prolactin (dose-dependent)
  • Tingling or numbness at injection site
  • Potential blood sugar effects
  • Significant cortisol and prolactin elevation (more than Ipamorelin)
  • Water retention
  • Increased appetite
  • Desensitization with prolonged use
  • Limited long-term human safety data
Regulatory Status
Unregulated

Not FDA-approved. Available as a research chemical. Pralmorelin (the INN name) has been studied clinically in Japan for GH deficiency diagnosis but has no approved therapeutic indication in the US.

Category 1

Reclassified to Category 1 in February 2026 as part of the HHS announcement restoring compounding access. Not affected by the April 15, 2026 Category 2 removal action. Available through licensed 503A compounding pharmacies with a physician prescription.

This comparison is for educational purposes only and does not constitute medical advice. Always consult a qualified healthcare professional before starting any peptide therapy.