Compare Peptides

Select any two compounds for a side-by-side comparison of mechanism, uses, risks, and FDA regulatory status.

Popular comparisons

Tirzepatide

Mounjaro, Zepbound

FDA Approved
GLP-1/GIP Dual Agonist

Retatrutide

LY3437943, Eli Lilly Triple Agonist

Investigational
GLP-1/GIP/Glucagon Triple Agonist
Overview

A dual GIP and GLP-1 receptor agonist developed by Eli Lilly. Represents the next generation of incretin-based therapies with potentially superior efficacy to semaglutide for weight loss.

An investigational triple-agonist peptide developed by Eli Lilly that targets GLP-1, GIP, and glucagon receptors simultaneously. Phase 3 clinical trials are underway, with early results showing unprecedented weight loss efficacy.

Mechanism of Action

Activates both GIP (glucose-dependent insulinotropic polypeptide) and GLP-1 receptors, producing enhanced insulin secretion, appetite suppression, and metabolic improvements beyond what single-agonist drugs achieve.

Activates three metabolic hormone receptors: GLP-1 (appetite suppression, insulin secretion), GIP (enhanced insulin response, fat metabolism), and glucagon (increased energy expenditure, fat oxidation). The triple mechanism may produce greater weight loss than dual agonists.

Common Uses
  • Weight management
  • Type 2 diabetes treatment
  • Metabolic health improvement
  • Weight management (investigational)
  • Type 2 diabetes (investigational)
  • Metabolic syndrome (investigational)
Known Risks
  • GI side effects (nausea, diarrhea, vomiting)
  • Pancreatitis risk
  • Injection site reactions
  • Potential thyroid concerns
  • Still in clinical trials — full safety profile unknown
  • GI side effects (nausea, diarrhea, vomiting) reported in trials
  • Not yet approved for any indication
  • Long-term effects unknown
Regulatory Status
FDA Approved

FDA-approved as Mounjaro (diabetes, 2022) and Zepbound (weight management, 2023).

Investigational

Currently in Phase 3 clinical trials. Phase 2 results showed up to 24% body weight loss at 48 weeks. FDA approval timeline uncertain but potentially 2027-2028.

This comparison is for educational purposes only and does not constitute medical advice. Always consult a qualified healthcare professional before starting any peptide therapy.