Compare Peptides

Select any two compounds for a side-by-side comparison of mechanism, uses, risks, and FDA regulatory status.

Popular comparisons

Dulaglutide

Trulicity

FDA Approved
GLP-1 Agonist

Exenatide

Byetta, Bydureon

FDA Approved
GLP-1 Agonist
Overview

A once-weekly GLP-1 receptor agonist FDA-approved for type 2 diabetes and cardiovascular risk reduction. Developed by Eli Lilly as a predecessor to tirzepatide. One of the most prescribed GLP-1 agonists globally.

The first GLP-1 receptor agonist approved by the FDA, originally derived from Gila monster saliva. Available in twice-daily (Byetta) and once-weekly (Bydureon) formulations. Paved the way for semaglutide and tirzepatide.

Mechanism of Action

A GLP-1 analog fused to a modified IgG4 Fc fragment, extending its half-life to approximately 5 days. Activates GLP-1 receptors to stimulate insulin secretion, suppress glucagon, slow gastric emptying, and reduce appetite.

Synthetic version of exendin-4, a peptide found in Gila monster venom that shares 53% homology with human GLP-1 but resists DPP-4 degradation. Stimulates insulin secretion, suppresses glucagon, slows gastric emptying, and promotes satiety.

Common Uses
  • Type 2 diabetes
  • Cardiovascular risk reduction
  • Moderate weight loss
  • Blood sugar regulation
  • Type 2 diabetes
  • Blood sugar regulation
  • Modest weight loss
Known Risks
  • GI side effects (nausea, diarrhea, vomiting)
  • Pancreatitis (rare)
  • Thyroid C-cell tumors (animal studies)
  • Injection site reactions
  • Hypoglycemia when combined with insulin
  • Nausea (common, especially initially)
  • Pancreatitis (rare)
  • Injection site nodules (Bydureon)
  • Renal impairment
  • Thyroid C-cell tumors (animal studies)
Regulatory Status
FDA Approved

FDA-approved as Trulicity (2014) for type 2 diabetes and cardiovascular risk reduction (REWIND trial). Once-weekly injection via single-dose pen. One of the top-selling GLP-1 drugs globally.

FDA Approved

FDA-approved as Byetta (2005, twice daily) and Bydureon (2012, once weekly). The first-in-class GLP-1 agonist. Largely superseded by semaglutide for new prescriptions but still widely used.

This comparison is for educational purposes only and does not constitute medical advice. Always consult a qualified healthcare professional before starting any peptide therapy.